The mechanism of allosteric coupling in choline kinase a1 revealed by a rationally designed inhibitor
External Resource: Annotation
Domain Annotation: SCOP2 Classification SCOP2 Database Homepage
Chains | Type | Family Name | Domain Identifier | Family Identifier | Provenance Source (Version) |
A | SCOP2 Family | Choline kinase | 8085226 | 4003732 | SCOP2 (2022-06-29) |
A | SCOP2 Superfamily | Protein kinase-like (PK-like) | 8085227 | 3000066 | SCOP2 (2022-06-29) |
B | SCOP2B Superfamily | Protein kinase-like (PK-like) | 8085227 | 3000066 | SCOP2B (2022-06-29) |
Chains | Family Name | Domain Identifier | Architecture | Possible Homology | Homology | Topology | Family | Provenance Source (Version) |
A | Fructosamin_kin | e3zm9A1 | A: a+b complex topology | X: Protein kinase/SAICAR synthase/ATP-grasp (From Homology) | H: Protein kinase/SAICAR synthase/ATP-grasp | T: Protein kinase | F: Fructosamin_kin | ECOD (1.6) |
B | Fructosamin_kin | e3zm9B2 | A: a+b complex topology | X: Protein kinase/SAICAR synthase/ATP-grasp (From Homology) | H: Protein kinase/SAICAR synthase/ATP-grasp | T: Protein kinase | F: Fructosamin_kin | ECOD (1.6) |
Chains | Polymer | Molecular Function | Biological Process | Cellular Component |
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| CHOLINE KINASE ALPHA | | | |
Chains | Drug Target   | Associated Disease |
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| Pharos:  P35790 | |